AZ10417808 is a selective non-peptide inhibitor of caspase-3 (Ki = 247 nM); displays > 40-fold selectivity over caspases 1, 2, 6, 7 and 8 (Ki > 10 μM). Completely blocks staurosporine-induced intracellular DEVDase activity in SH-SY5Y cells (IC₅₀ = 14

Item Number: BIOV2786-1
Unit of Measure: 1 MG
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94.60 CHF 94.60000000000001 CHF 94.60 CHF

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    Manufacturer: BIOVISION
    Manufacturer Number: 2786-1
    Storage Temperature: Freezer (-20)

    AZ10417808 is a selective non-peptide inhibitor of caspase-3 (Ki = 247 nM); displays > 40-fold selectivity over caspases 1, 2, 6, 7 and 8 (Ki > 10 μM). Completely blocks staurosporine-induced intracellular DEVDase activity in SH-SY5Y cells (IC₅₀ = 14