GSK-2656157 is a potent, selective and ATP-competitive inhibitor of PERK (protein kinase R-like ER kinase) enzyme activity with an I C₅₀ of 0.9 nM; displays high selectivity for PERK against a panel of 300 kinases (IC₅₀>100 nM).
Item Number: BIOV9466-5
Unit of Measure: 5 MG
Manufacturer: BIOVISION
Manufacturer Number: 9466-5
Storage Temperature: Freezer (-20)
GSK-2656157 is a potent, selective and ATP-competitive inhibitor of PERK (protein kinase R-like ER kinase) enzyme activity with an I C₅₀ of 0.9 nM; displays high selectivity for PERK against a panel of 300 kinases (IC₅₀>100 nM).
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