Potent, cell permeable inhibitor of PHD2 (IC50 = 21 nM) with over 100-fold selectivity compared to inhibition of JMJD2A, JMJD2C, JMJ D2E, JMJD3, or the 2OG oxygenase FIH (IC50s > 100 μM), UoM: 1 * 25 mg
Item Number: CAYM11573-25
Unit of Measure: 25 MG
Manufacturer: CAYMAN
Manufacturer Number: 11573-25
Storage Temperature: Freezer (-20)
Potent, cell permeable inhibitor of PHD2 (IC50 = 21 nM) with over 100-fold selectivity compared to inhibition of JMJD2A, JMJD2C, JMJ D2E, JMJD3, or the 2OG oxygenase FIH (IC50s > 100 μM), UoM: 1 * 25 mg
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