CB5083 is a potent, ATP-competitive, D2-selective, p97 inhibitor (IC₅₀ = 11 nM). In xenograft models, CB-5083 causes modulation of k ey p97-related pathways, induces apoptosis, and has antitumor activity in a broad range of both hematological and sol

Numéro d'article : BIOVB1032-5
Unité de mesure : 5 MG
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    Numéro CAS : 1542705-92-9
    Fabricant : BIOVISION
    Numéro du fabricant : B1032-5
    Formule chimique : C24H23N5O2
    Température de stockage : Freezer (-20)

    CB5083 is a potent, ATP-competitive, D2-selective, p97 inhibitor (IC₅₀ = 11 nM). In xenograft models, CB-5083 causes modulation of k ey p97-related pathways, induces apoptosis, and has antitumor activity in a broad range of both hematological and sol