BLU9931 is a potent and irreversible small-molecule inhibitor of FGFR4. It potently inhibits FGFR4 activity (IC₅₀ = 3 nM), but only weakly inhibits FGFR1 (IC₅₀ = 591 nM), FGFR2 (IC₅₀ = 493 nM), and FGFR3 (IC₅₀ = 150 nM) activity.

Numero articolo: BIOV9639-25
Unità di misura: 25 MG
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    Produttore: BIOVISION
    Numero del produttore: 9639-25
    Temperatura di stoccaggio: Freezer (-20)

    BLU9931 is a potent and irreversible small-molecule inhibitor of FGFR4. It potently inhibits FGFR4 activity (IC₅₀ = 3 nM), but only weakly inhibits FGFR1 (IC₅₀ = 591 nM), FGFR2 (IC₅₀ = 493 nM), and FGFR3 (IC₅₀ = 150 nM) activity.